Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse
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DOI: 10.1021/acs.jmedchem.5c00395
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c00395
其他信息:
出版社: American Chemical Society (ACS)
作者: Anthony K. Edmonds; Dimitrios-Ilias Balourdas; Graham P. Marsh; Robert Felix; Bradley Brasher; Jeff Cooper; Cari Graber-Feesl; Madhu Kollareddy; Karim Malik; Helen Stewart; Timothy J. T. Chevassut; Ella Lineham; Simon Morley; Oleg Fedorov; James Bennett; Mohan B. Rajasekaran; Samuel Ojeda; Drew A. Harrison; Christopher J. Ott; Andreas C. Joerger; Hannah J. Maple; John Spencer
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c00395